Detalles de la búsqueda
1.
In silico Design, Synthesis and Biological Evaluation of Novel Thieno[3,2-d]pyrimidine Derivatives for Cancer Therapy - A Preliminary Study on the Inhibitory Potential towards ATR Kinase Domain and PIKK Family.
Chem Biodivers
; 21(3): e202302071, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38230843
2.
Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies.
Bioorg Chem
; 138: 106621, 2023 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-37257407
3.
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors.
Int J Mol Sci
; 24(3)2023 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36769114
4.
Discovery of Novel EGFR Inhibitor Targeting Wild-Type and Mutant Forms of EGFR: In Silico and In Vitro Study.
Molecules
; 28(7)2023 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37049777
5.
New Bicyclic Pyridine-Based Hybrids Linked to the 1,2,3-Triazole Unit: Synthesis via Click Reaction and Evaluation of Neurotropic Activity and Molecular Docking.
Molecules
; 28(3)2023 Jan 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-36770592
6.
Synthesis of 1-Amino-3-oxo-2,7-naphthyridines via Smiles Rearrangement: A New Approach in the Field of Chemistry of Heterocyclic Compounds.
Int J Mol Sci
; 23(11)2022 May 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-35682584
7.
Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents.
Molecules
; 27(14)2022 Jul 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-35889508
8.
Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives.
Molecules
; 27(3)2022 Feb 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35164333
9.
Antibacterial activity of noscapine analogs.
Bioorg Med Chem Lett
; 43: 128055, 2021 07 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33892103
10.
Synthesis and antimicrobial activity of new 2-piperazin-1-yl-N-1,3-thiazol-2-ylacetamides of cyclopenta[c]pyridines and pyrano[3,4-c]pyridines.
Arch Pharm (Weinheim)
; 354(1): e2000208, 2021 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-33029832
11.
Chromene-Containing Aromatic Sulfonamides with Carbonic Anhydrase Inhibitory Properties.
Int J Mol Sci
; 22(10)2021 May 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-34064890
12.
Disruption of the Complex between GAPDH and Hsp70 Sensitizes C6 Glioblastoma Cells to Hypoxic Stress.
Int J Mol Sci
; 22(4)2021 Feb 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-33546324
13.
Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors.
Molecules
; 26(22)2021 Nov 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-34834114
14.
Synthesis and Neurotropic Activity of New Heterocyclic Systems: Pyridofuro[3,2-d]pyrrolo[1,2-a]pyrimidines, Pyridofuro[3,2-d]pyrido[1,2-a]pyrimidines and Pyridofuro[3',2':4,5]pyrimido[1,2-a]azepines.
Molecules
; 26(11)2021 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-34205930
15.
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials.
Mol Divers
; 24(1): 233-239, 2020 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-30949901
16.
5-(1H-Indol-3-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)alkancarboxylic Acids as Antimicrobial Agents: Synthesis, Biological Evaluation, and Molecular Docking Studies.
Molecules
; 25(8)2020 Apr 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-32340255
17.
Structure of Dirithromycin Bound to the Bacterial Ribosome Suggests New Ways for Rational Improvement of Macrolides.
Antimicrob Agents Chemother
; 63(6)2019 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-30936109
18.
Madumycin II inhibits peptide bond formation by forcing the peptidyl transferase center into an inactive state.
Nucleic Acids Res
; 45(12): 7507-7514, 2017 Jul 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-28505372
19.
Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.
Molecules
; 24(19)2019 Oct 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-31590289
20.
Application of Docking Analysis in the Prediction and Biological Evaluation of the Lipoxygenase Inhibitory Action of Thiazolyl Derivatives of Mycophenolic Acid.
Molecules
; 23(7)2018 Jul 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-29970872